Sfoglia per Autore
Synthesis and antimycobacterial activity of 1,3,4-oxadiazol-2-one derivatives.
2007-01-01 Mamolo, MARIA GRAZIA; Laurini, Erik; Vio, Luciano; G., Scialino; Banfi, Elena; Zampieri, Daniele
3-Piperidin-4-yl-methyl-3H-benzoxazol-2-one derivatives as sigma ligands.
2007-01-01 Mamolo, MARIA GRAZIA; Zampieri, Daniele; Laurini, Erik; Vio, Luciano; S., Collina; D., Rossi; O., Azzolina; Florio, Chiara; C., Zanette
Synthesis and antifungal activity of new N-[1-aryl-2-(1H-imidazol-1-yl and 1H-1,2,4-triazol-1-yl)-1-ethylidene]-N'-phenylhydrazine derivatives.
2007-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Vio, Luciano; G., Scialino; Banfi, Elena
Antifungal and antimycobacterial activity of 1-(3,5-diaryl-4,5-dihydro-1H-pyrazol-4-yl)-1H-imidazole derivatives.
2008-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Scialino, Giuditta; Banfi, Elena; Vio, Luciano
A new class of substituted benzo[d]oxazole-2(3H)-one derivatives as sigma1 ligands.
2008-01-01 Mamolo, MARIA GRAZIA; Zampieri, Daniele; Laurini, Erik; Vio, Luciano; S., Collina; O., Azzolina; D., Rossi; Florio, Chiara; C., Zanette
Antimycobacterial activity of new 3,5-disubstituted 1,3,4-oxadiazol-2(3H)-one derivatives. Molecular modeling investigations
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Fermeglia, Maurizio; Posocco, Paola; Pricl, Sabrina; Banfi, Elena; Scialino, Giuditta; Vio, Luciano
2-Aryl-3-(1H-azol-1-yl)-1H-indole derivatives: a new class of antimycobacterial compounds. Convetional heating in comparison with MW-assisted synthesis.
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Scialino, Giuditta; Banfi, Elena; Vio, Luciano
Substituted benzo[d]oxazol-2(3H)-one derivatives with preference for the σ1 binding site
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Zanette, Caterina; Florio, Chiara; Collina, S; Rossi, D; Azzolina, O; Vio, Luciano
Synthesis, biological evaluation, and three-dimensional in silico pharmacophore model for sigma1 receptor ligand based on a series of benzo[d]oxazol-2(3H)-one derivatives
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Florio, Chiara; Zanette, Caterina; Fermeglia, Maurizio; Posocco, Paola; Paneni, Maria Silvia; Pricl, Sabrina; Vio, Luciano
When virtual and real meet: computational/experimental evidences for designing efficient nanovectors for siRNA/DNA delivery
2010-01-01 Pricl, Sabrina; Posocco, Paola; Laurini, Erik; Fermeglia, Maurizio; Karatasos, K.; Peng, L.; Smith, D. K.
The Novel BCR-ABL1 V304D Mutation Induces Pan-Tyrosine Kinase Inhibitor Resistance by a Unique Kinase Lateral Escape Mechanism and Is Associated with Very Poor Prognosis In Patients (PTS) with Chronic Myeloid Leukemia (CML)
2010-01-01 Pricl, Sabrina; D. L., Gibbons; Posocco, Paola; Laurini, Erik; Fermeglia, Maurizio; H. M., Kantarjian; M., Talpaz; J., Cortes; M., Young; H., Sun; L. F., Peterson; N., Donato; A., Quintas Cardama
A 3D-Pharmacophore Model for σ2 Receptors Based on a Series of Substituted Benzo[d]oxazol-2(3H)-one Derivatives
2010-01-01 Laurini, Erik; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Vio, Luciano; Zanette, Caterina; Florio, Chiara; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina
SYNTHESIS, MOLECULAR MODELING AND EXPERIMENTALACTIVITY OF SOME NEW ACETAMIDE, BENZAMIDE ANDPHENYLMETHANONE DERIVATIVES AS SIGMA LIGANDS.
2010-01-01 Laurini, Erik; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Vio, Luciano; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina; Zanette, Caterina; Florio, Chiara
In Silico modelling of Sensitivity to Novel Tyrosine Kinase Inhibitors of Highly Resistant Single and Polymutant BCR-ABL1
2010-01-01 Pricl, Sabrina; Gibbons, Dl; Posocco, Paola; Laurini, Erik; Fermeglia, Maurizio; Kantarjian, Hm; Talpaz, M; Cortes, J; Donato, N; Quintas Cardama, A.
Synergistic experimental/computational studies on arylazoenamine derivatives that target the bovine viral diarrhea virus RNA-dependent RNA polymerase
2010-01-01 Gabriele, Giliberti; Cristina, Ibba; Esther, Marongiu; Roberta, Loddo; Michele, Tonelli; Vito, Boido; Laurini, Erik; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina
Nanozapped! DNA, siRNA, and their dendritic nanovectors: a combined in silico/in vitro/in vivo approach
2011-01-01 Dal Col, V; Laurini, Erik; Posocco, Paola; Pricl, Sabrina; Liu, Xx; Peng, L; Jones, Sp; Barnard, A; Smith, Dk
The long and winding road of the c-Kit juxtamembrane domain
2011-01-01 V., Dal Col; Laurini, Erik; Pricl, Sabrina; Posocco, Paola; M. A., Pierotti; P., Casali; S., Pilotti; E., Tamborini
Overview on σ1 receptor: a 3D homology model to solve a part of the enigma.
2011-01-01 Laurini, Erik; V., Dal Col; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Posocco, Paola; Pricl, Sabrina; Vio, Luciano
In silico exploration of the Embryonic Lethal Abnormal Vision protein-mRNA interaction followed by in vitro bioassays for the identification of peptides potentially useful in neurodegenerative diseases treatment
2011-01-01 Carnevale Baraglia, A; Amadio, M; Pascale, A; Govoni, S; Laurini, Erik; Pricl, Sabrina; Rossi, D; Azzolina, O; Collina, S.
The sigma-enigma. A multistep homology modeling of sigma1 receptors
2011-01-01 Laurini, Erik; Dal Col, V; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Posocco, Paola; Vio, Luciano; Pricl, Sabrina
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