Sfoglia per Autore
Through the open door: Preferential binding of dasatinib to the active form of BCR-ABL unveiled by in silico experiments
2013-01-01 Laurini, Erik; Posocco, Paola; Fermeglia, Maurizio; Gibbons, Dl; Quintás Cardama, A; Pricl, Sabrina
Novel inhibitors of signal transducer and activator of transcription 3 (STAT3) show potent activity in cell cultures and tumor xenografts.
2014-01-01 Genini, Davide; Brambilla, Lara; Laurini, Erik; Civenni, Gianluca; Pinton, Sandra; Sarti, Manuela; Garcia Escudero, Ramon; Perez, Laurent; Carbone, Giuseppina M.; Pricl, Sabrina; Catapano, Carlo V.
Molecular dynamics reveal BCR-ABL1 polymutants as a unique mechanism of resistance to PAN-BCR-ABL1 kinase inhibitor therapy
2014-01-01 Gibbons, Dl; Pricl, Sabrina; Posocco, Paola; Laurini, Erik; Fermeglia, Maurizio; Sun, H; Talpaz, M; Donato, N; Quintás Cardama, A.
Copper(ii) binding to flexible triethanolamine-core PAMAM dendrimers: a combined experimental/in silico approach
2014-01-01 Maria Francesca, Ottaviani; Michela, Cangiotti; Alberto, Fattori; Concetta, Coppola; Posocco, Paola; Laurini, Erik; Xiaoxuan, Liu; Cheng, Liu; Fermeglia, Maurizio; Ling, Peng; Pricl, Sabrina
Synthesis, pharmacological evaluation and σ1 receptor interaction analysis of hydroxyethyl substituted piperazines
2014-01-01 Frauke, Weber; Steffi, Brune; Katharina, Korpis; Patrick J., Bednarski; Laurini, Erik; DAL COL, Valentina; Pricl, Sabrina; Dirk, Schepmann; Bernhard, Wünsch
Identification, pharmacological evaluation and binding mode analysis of novel chromene and chromane based σ1 receptor ligands
2014-01-01 Laurini, Erik; Dipak, Harel; Marson, Domenico; Dirk, Schepmann; Thomas J., Schmidt; Pricl, Sabrina; Bernhard, Wünsch
The Sigma Enigma:In Vitro/in SilicoSite-Directed Mutagenesis Studies Unveil σ1Receptor Ligand Binding
2014-01-01 S., Brune; D., Schepmann; K. H., Klempnauer; Marson, Domenico; DAL COL, Valentina; Laurini, Erik; Fermeglia, Maurizio; B., Wünsch; Pricl, Sabrina
Mimicking the 2-oxoglutaric acid signalling function using molecular probes: insights from structural and functional investigations
2014-01-01 Yang, Wang; Xinjun, Liu; Laurini, Erik; Posocco, Paola; Fabio, Ziarelli; Fermeglia, Maurizio; Fanqi, Qu; Pricl, Sabrina; Cheng Cai, Zhang; Ling, Peng
Synthesis and receptor binding studies of some new arylcarboxamide derivatives as sigma-1 ligands
2014-01-01 Zampieri, Daniele; Laurini, Erik; Vio, Luciano; Golob, Samuel; Fermeglia, Maurizio; Pricl, Sabrina; Mamolo, MARIA GRAZIA
Benzoxazinones and correlated scaffolds linked to benzylamino moieties through a butylene spacer. New sigma receptor ligands
2015-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Vio, Luciano; Laurini, Erik; Pricl, Sabrina; Fermeglia, Maurizio; Schepmann, D.; Wünsch, B.
A methodology for the sustainability evaluation of industrial pharmaceutical processes
2015-01-01 Mio, Andrea; Laurini, Erik; Pricl, Sabrina; Fermeglia, Maurizio
Still looking for the magic spot: dispersing modified Fe2O3 in lamellar PS-PMMA diblock copolymer by vapor-annealing deposition
2015-01-01 Posocco, Paola; Mohamed, Y.; Barandiaran, I.; Zweyer, Marina; Baldini, Giovanna; Laurini, Erik; Fermeglia, Maurizio; Kortaberria, G.; Pricl, Sabrina
Of (computers and cells) mice and men: Integration of Simulations and Experiments in biomedical sciences.
2015-01-01 Laurini, Erik; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina
Of (computers, cells) mice and men: Integration of simulations and experiments in molecular medicine
2015-01-01 Pricl, Sabrina; Fermeglia, Maurizio; Posocco, Paola; Marson, Domenico; Laurini, Erik
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives
2015-01-01 Briguglio, Irene; Loddo, Roberta; Laurini, Erik; Fermeglia, Maurizio; Piras, Sandra; Corona, Paola; Giunchedi, Paolo; Gavini, Elisabetta; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; La Colla, Paolo; Pricl, Sabrina; Carta, Antonio
MoDeNa: Modeling of morphology Development of micro and Nano Structures
2015-01-01 Laurini, Erik; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina
Improving selectivity preserving affinity: New piperidine-4-carboxamide derivatives as effective sigma-1-ligands
2015-01-01 Zampieri, Daniele; Laurini, Erik; Vio, Luciano; Fermeglia, Maurizio; Pricl, Sabrina; Wünsch, Bernhard; Schepmann, Dirk; Mamolo, MARIA GRAZIA
Smoothened (SMO) receptor mutations dictate resistance to vismodegib in basal cell carcinoma
2015-01-01 Pricl, Sabrina; Barbara, Cortelazzi; DAL COL, Valentina; Marson, Domenico; Laurini, Erik; Fermeglia, Maurizio; Lisa, Licitra; Silvana, Pilotti; Paolo, Bossi; Federica, Perrone
A step forward in the sigma enigma: a role for chirality in the sigma1 receptor–ligand interaction?
2015-01-01 Daniela, Rossi; Annamaria, Marra; Marta, Rui; Laurini, Erik; Fermeglia, Maurizio; Pricl, Sabrina; Dirk, Schepmann; Bernhard, Wuensch; Marco, Peviani; Daniela, Curti; Simona, Collina
Cationic carbosilane dendrimers and oligonucleotide binding: an energetic affair
2015-01-01 Marson, Domenico; Laurini, Erik; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina
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