PRENCIPE, FILIPPO
PRENCIPE, FILIPPO
Dipartimento di Scienze Chimiche e Farmaceutiche
Ricercatori a tempo determinato
3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
2018-01-01 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
7-Amino-[1,2,4]triazolo[1,5-a][1,3,5]triazines as CK1δ inhibitors: Exploring substitutions at the 2 and 5-positions
2024-01-01 Grieco, Ilenia; Bassani, Davide; Trevisan, Letizia; Salmaso, Veronica; Cescon, Eleonora; Prencipe, Filippo; Da Ros, Tatiana; Martinez-Gonzalez, Loreto; Martinez, Ana; Spalluto, Giampiero; Moro, Stefano; Federico, Stephanie
[1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell Lines
2023-01-01 Federico, S.; Persico, M.; Trevisan, L.; Biasinutto, C.; Bolcato, G.; Salmaso, V.; Da Ros, T.; Gianferrara, T.; Prencipe, F.; Kachler, S.; Klotz, K. -N.; Pacor, S.; Moro, S.; Spalluto, G.
Adenosine Receptor Ligands, Probes, and Functional Conjugates: A 20-Year History of Pyrazolo[4,3-e][1,2,4]Triazolo[1,5-c]Pyrimidines (PTP)
2023-01-01 Prencipe, F.; Da Ros, T.; Cescon, E.; Grieco, I.; Persico, M.; Spalluto, G.; Federico, S.
Allantodapsone is a Pan-Inhibitor of Staphylococcus aureus Adhesion to Fibrinogen, Loricrin, and Cytokeratin 10
2022-01-01 Prencipe, Filippo; Alsibaee, Aishah; Khaddem, Zainab; Norton, Padraig; Towell, Aisling M; Ali, Afnan F M; Reid, Gerard; Fleury, Orla M; Foster, Timothy J; Geoghegan, Joan A; Rozas, Isabel; Brennan, Marian P
Apoptosis Pathways Triggered by a Potent Antiproliferative Hybrid Chalcone on Human Melanoma Cells
2021-01-01 Rodríguez, Irene; Saavedra, Ester; del Rosario, Henoc; Perdomo, Juan; Quintana, José; Prencipe, Filippo; Oliva, Paola; Romagnoli, Romeo; Estévez, Francisco
Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis
2022-01-01 Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Germanò, Maria Paola; De Luca, Laura; Ricci, Federico; Corallo, Diana; Aveic, Sanja; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3’,4’,5’-Trimethoxyphenyl)-2-Aryl-1H-Imidazole
2016-01-01 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; AGHAZADEH TABRIZI, Mojgan; Lopez Cara, Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro .
Design, synthesis and antiproliferative activity of novel heterobivalent hybrids based on imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b][1,3]thiazole scaffolds
2015-01-01 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Balzarini, Jan; Liekens, Sandra; Estévez, Francisco
Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization
2020-01-01 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Kimatrai Salvador, Maria; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Viola, Giampietro; Bortolozzi, Roberta; Persoons, Leentje; Balzarini, Jan; Liekens, Sandra; Schols, Dominique
Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents
2017-01-01 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Bortolozzi, Roberta; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro
Design, Synthesis and Biological Evaluation of Arylcinnamide Hybrid Derivatives as Novel Anticancer Agents
2014-01-01 Romagnoli, Romeo; Baraldi, Pier Giovanni; Maria Kimatrai, Salvador; Mariem, Chayah; M., Encarnacion Camacho; Prencipe, Filippo; Ernest, Hamel; Francesca, Consolaro; Giuseppe, Basso; Giampietro, Viola
Design, Synthesis and Biological Investigation of 2-Anilino Triazolopyrimidines as Tubulin Polymerization Inhibitors with Anticancer Activities
2022-01-01 Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Budassi, Federica; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Manfreda, Lorenzo; Mariotto, Elena; Bortolozzi, Roberta; Viola, Giampietro
Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors
2019-01-01 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Schiaffino Ortega, Santiago; Chayah, Mariem; Kimatrai Salvador, Maria; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Mattiuzzo, Elena; Viola, Giampietro
Design, synthesis, in vitro, and in vivo anticancer and antiangiogenic activity of novel 3-arylaminobenzofuran derivatives targeting the colchicine site on tubulin
2015-01-01 Romagnoli, Romeo; Baraldi, Pier Giovanni; Salvador, Maria Kimatrai; Prencipe, Filippo; Lopez Cara, Carlota; Schiaffino Ortega, Santiago; Brancale, Andrea; Hamel, Ernest; Castagliuolo, Ignazio; Mitola, Stefania; Ronca, Roberto; Bortolozzi, Roberta; Porcù, Elena; Basso, Giuseppe; Viola, Giampietro
Disclosing the Preferential Mercury Chelation by SeCys Containing Peptides over Their Cys Analogues
2023-01-01 Bernabeu de Maria, M.; Tesauro, D.; Prencipe, F.; Saviano, M.; Messori, L.; Enjalbal, C.; Lobinski, R.; Ronga, L.
Forward Precision Medicine: Micelles for Active Targeting Driven by Peptides
2021-01-01 Prencipe, Filippo; Diaferia, Carlo; Rossi, Filomena; Ronga, Luisa; Tesauro, Diego
Gaucher Disease: A Glance from a Medicinal Chemistry Perspective
2024-01-01 Prencipe, Filippo; Barzan, Chiara; Savian, Chiara; Spalluto, Giampiero; Carosati, Emanuele; DE AMICI, Marco; Mosconi, Giorgio; Gianferrara, Teresa; Federico, Stephanie; DA ROS, Tatiana
New Insights into the Behavior of NHC-Gold Complexes in Cancer Cells
2023-01-01 Augello, Giuseppa; Azzolina, Antonina; Rossi, Filomena; Prencipe, Filippo; Mangiatordi, Giuseppe Felice; Saviano, Michele; Ronga, Luisa; Cervello, Melchiorre; Tesauro, Diego
Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation
2016-01-01 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Lopez Cara, Carlota; Rondanin, Riccardo; Simoni, Daniele; Hamel, Ernest; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Tolomeo, Manlio