Sfoglia per Autore
2-Aryl-3-(1H-azol-1-yl)-1H-indole derivatives: a new class of antimycobacterial compounds. Convetional heating in comparison with MW-assisted synthesis.
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Scialino, Giuditta; Banfi, Elena; Vio, Luciano
Synthesis and antimycobacterial activity of some new pyridine-2-carboxamidrazone derivatives.
2009-01-01 Zampieri, Daniele; E., Laurini; Mamolo, MARIA GRAZIA; L., Vio
New prospective in the design and in the synthesis of new sigma ligands: computational approach and classic way.
2009-01-01 E., Laurini; Mamolo, MARIA GRAZIA; Zampieri, Daniele; S., Collina; D., Rossi; L., Vio
FROM 3D PHARMACOPHORE MODEL TO SYNTHESIS: A NEW SERIES OF 1-BENZYL-PIPERIDINE-4-CARBOXYLIC ACID BENZYLAMIDE DERIVATIVES AS NEW s1 LIGANDS.
2009-01-01 E., Laurini; Mamolo, MARIA GRAZIA; Zampieri, Daniele; C., Florio; C., Zanette; Pricl, Sabrina; Fermeglia, Maurizio; L., Vio
Substituted benzo[d]oxazol-2(3H)-one derivatives with preference for the σ1 binding site
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Zanette, Caterina; Florio, Chiara; Collina, S; Rossi, D; Azzolina, O; Vio, Luciano
Synthesis, biological evaluation, and three-dimensional in silico pharmacophore model for sigma1 receptor ligand based on a series of benzo[d]oxazol-2(3H)-one derivatives
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Florio, Chiara; Zanette, Caterina; Fermeglia, Maurizio; Posocco, Paola; Paneni, Maria Silvia; Pricl, Sabrina; Vio, Luciano
Antimycobacterial activity of new 3,5-disubstituted 1,3,4-oxadiazol-2(3H)-one derivatives. Molecular modeling investigations
2009-01-01 Zampieri, Daniele; Mamolo, MARIA GRAZIA; Laurini, Erik; Fermeglia, Maurizio; Posocco, Paola; Pricl, Sabrina; Banfi, Elena; Scialino, Giuditta; Vio, Luciano
SYNTHESIS, MOLECULAR MODELING AND EXPERIMENTALACTIVITY OF SOME NEW ACETAMIDE, BENZAMIDE ANDPHENYLMETHANONE DERIVATIVES AS SIGMA LIGANDS.
2010-01-01 Laurini, Erik; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Vio, Luciano; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina; Zanette, Caterina; Florio, Chiara
Design, synthesis and SAR analysis of novel selective sigma1 ligands (Part 2)
2010-01-01 D., Rossi; M., Urbano; A., Pedrali; M., Serra; Zampieri, Daniele; Mamolo, MARIA GRAZIA; C., Laggner; Zanette, Caterina; Florio, Chiara; D., Schepmann; B., Wuensch; O., Azzolina; Collina, Simona
A 3D-Pharmacophore Model for σ2 Receptors Based on a Series of Substituted Benzo[d]oxazol-2(3H)-one Derivatives
2010-01-01 Laurini, Erik; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Vio, Luciano; Zanette, Caterina; Florio, Chiara; Posocco, Paola; Fermeglia, Maurizio; Pricl, Sabrina
Analisi Farmaceutica Qualitativa
2011-01-01 Mamolo, MARIA GRAZIA; Zampieri, Daniele; Vio, Luciano
Overview on σ1 receptor: a 3D homology model to solve a part of the enigma.
2011-01-01 Laurini, Erik; V., Dal Col; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Posocco, Paola; Pricl, Sabrina; Vio, Luciano
The sigma-enigma. A multistep homology modeling of sigma1 receptors
2011-01-01 Laurini, Erik; Dal Col, V; Zampieri, Daniele; Mamolo, MARIA GRAZIA; Posocco, Paola; Vio, Luciano; Pricl, Sabrina
New alkylacetamide derivatives as new sigma ligands.
2011-01-01 Zampieri, Daniele; Laurini, Erik; Mamolo, MARIA GRAZIA; Florio, Chiara; Vio, Luciano
Design, synthesis and biological profile of new piperidine-4-carboxamide as effective sigma ligands
2011-01-01 Laurini, Erik; Mamolo, MARIA GRAZIA; Zampieri, Daniele; Vio, Luciano; Florio, Chiara
Homology Model and Docking-Based Virtual Screening for Ligands of the σ1 Receptor
2011-01-01 Laurini, Erik; DAL COL, Valentina; Mamolo, MARIA GRAZIA; Zampieri, Daniele; Posocco, Paola; Fermeglia, Maurizio; Vio, Luciano; Pricl, Sabrina
The sigma enigma. 3D homology modeling, computer-assisted drug design, 3D pharmacophore-guided docking, MM/PBSA scoring, in silico/in vitro alanine scanning mutagenesis, and functional assay to unveil the sigma-1 receptor hidden secrets.
2012-01-01 Mamolo, MARIA GRAZIA; Laurini, Erik; V., Dal Col; D., Marson; Zampieri, Daniele; Vio, Luciano; Pricl, Sabrina
Another Brick in the Wall. Validation of the σ1Receptor 3D Model by Computer-Assisted Design, Synthesis, and Activity of New σ1Ligands
2012-01-01 Laurini, Erik; Marson, Domenico; Valentina Dal Col, ; Fermeglia, Maurizio; Mamolo, MARIA GRAZIA; Zampieri, Daniele; Vio, Luciano; Pricl, Sabrina
New heterocyclic derivatives of benzylpiperidin-4-yl methyl and benzyl(methyl)aminobutyl sequences as sigma ligands.
2013-01-01 Zampieri, Daniele; Laurini, Erik; A., Sveronis; Vio, Luciano; Mamolo, MARIA GRAZIA
New heterocyclic derivatives of benzylpiperidin-4-yl methyl and benzyl(methyl)aminobutyl sequences as sigma ligands.
2013-01-01 Zampieri, Daniele; Laurini, Erik; Pricl, Sabrina; Vio, Luciano; Mamolo, MARIA GRAZIA
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