Sfoglia per Autore
Exploring Directionality of 5-Substitutions in a New Series of 5-Alkyamino-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a Strategy to Design Novel Human A3 Adenosine Receptors Antagonists.
2012-01-01 Federico, Stephanie; Ciancetta, Antonella; Paoletta, Silvia; Pastorin, Giorgia; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
Structural Investigations on a Novel Class of [1,2,4]Triazolo[1,5-c]pyrimidines as Adenosine Receptor Antagonists.
2012-01-01 Federico, Stephanie; Paoletta, Silvia; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
Simplification of Pyrazolo-triazolo-pyrimidine Nucleus for Searching New Adenosine Receptor Antagonists.
2012-01-01 Spalluto, Giampiero; Federico, Stephanie; Pastorin, Giorgia; Paoletta, Silvia; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano
Fluorescent ligands for the A3 adenosine receptor.
2012-01-01 Federico, Stephanie; Paoletta, Silvia; Kozma, Eszter; Kumar, T. Santhosh; Phan, Khai; Gao, Zhan Guo; Jacobson, Kenneth A.; Moro, Stefano; Spalluto, Giampiero
[1,2,4]Triazolo[1,5-c]pyrimidine Nucleus as Adenosine Receptor Antagonists: Shift in Selectivity from A2A to A3 Adenosine Receptors.
2012-01-01 Federico, Stephanie; Ciancetta, Antonella; Paoletta, Silvia; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
FLUORESCENT ANTAGONISTS OF THE A3 ADENOSINE RECEPTOR
2013-01-01 Kenneth A., Jacobson; Santosh Kumar, Thatikonda; Eszter Erika, Kozma; Spalluto, Giampiero; Stefano, Moro; Federico, Stephanie
Revisiting a Receptor-Based Pharmacophore Hypothesis for Human A2A Adenosine Receptor Antagonists
2013-01-01 Magdalena, Bacilieri; Antonella, Ciancetta; Silvia, Paoletta; Federico, Stephanie; Sandro, Cosconati; Barbara, Cacciari; Sabrina, Taliani; Federico Da, Settimo; Ettore, Novellino; Karl Norbert, Klotz; Spalluto, Giampiero; Stefano, Moro
The A3 adenosine receptor as multifaceted therapeutic Target: pharmacology, medicinal Chemistry, and In silico approaches
2013-01-01 Cheong, S. L.; Federico, Stephanie; Venkatesan, G.; Mandel, L.; Shao, Y. M.; Moro, S.; Spalluto, Giampiero; Pastorin, G.
Fluorescent ligands for adenosine receptors
2013-01-01 Eszter, Kozma; P., Suresh Jayasekara; Lucia, Squarcialupi; Silvia, Paoletta; Stefano, Moro; Federico, Stephanie; Spalluto, Giampiero; Kenneth A., Jacobson
8-(2-Furyl)adenine derivatives as A2A adenosine receptor ligands
2013-01-01 Diego Dal, Ben; Michela, Buccioni; Catia, Lambertucci; Ajiroghene, Thomas; Karl Norbert, Klotz; Federico, Stephanie; Barbara, Cacciari; Spalluto, Giampiero; Rosaria, Volpini
Revisiting a Receptor-Based Pharmacophore Hypothesis for Human A2A Adenosine Receptor Antagonists.
2013-01-01 Bacilieri, Magdalena; Ciancetta, Antonella; Paoletta, Silvia; Federico, Stephanie; Cosconati, Sandro; Cacciari, Barbara; Taliani, Sabrina; Settimo, Federico Da; Novellino, Ettore; Klotz, Karl Norbert; Spalluto, Giampiero; Moro, Stefano
1,2,4]Triazolo[1,5-c]pyrimidines as New Potent Human A3 Adenosine Receptor Antagonists.
2013-01-01 Spalluto, Giampiero; Federico, Stephanie; Ciancetta, Antonella; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano
Novel fluorescent hA3 adenosine receptor antagonists.
2013-01-01 Federico, Stephanie; Kozma, Eszter; Kumar, T. Santhosh; Jacobson, Kenneth A.; Moro, Stefano; Spalluto, Giampiero
[1,2,4]Triazolo[1,5-a][1,3,5]Triazine Derivatives as Antagonists for the Adenosine Receptors: a Preliminary Study on Affinity at the A3 Subtype
2013-01-01 Federico, Stephanie; Ciancetta, Antonella; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
N8-Isopentyl and N8-Phenylethyl Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine Derivatives as Adenosine Receptor Antagonists
2014-01-01 Federico, Stephanie; Redenti, Sara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
Scaffold decoration at positions 5 and 8 of 1,2,4-triazolo[1,5- c ]pyrimidines to explore the antagonist profiling on adenosine receptors: A preliminary structure-activity relationship study
2014-01-01 Federico, Stephanie; Ciancetta, Antonella; Porta, Nicola; Redenti, Sara; Pastorin, Giorgia; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
Discovery of simplified N2-substituted pyrazolo[3,4-d]pyrimidine derivatives as novel adenosine receptor antagonists: Efficient synthetic approaches, biological evaluations and molecular docking studies
2014-01-01 Gopalakrishnan, Venkatesan; Priyankar, Paira; Siew Lee, Cheong; Kosaraju, Vamsikrishna; Federico, Stephanie; Karl Norbert, Klotz; Spalluto, Giampiero; Giorgia, Pastorin
Conjugable A3 Adenosine Receptor Antagonists: Probing the 5 Position of the Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine Scaffold.
2014-01-01 Federico, Stephanie; Redenti, Sara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
CVT 6975-like Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine Derivatives: an Attempt towards A2B Adenosine Receptor Affinity.
2014-01-01 Redenti, Sara; Federico, Stephanie; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
[1,2,4]triazolo[1,5-c]pyrimidines as A(3) adenosine receptor antagonists
2014-01-01 Federico, Stephanie; Redenti, Sara; Ciancetta, Antonella; Cacciari, Barbara; Klotz, Karl Norbert; Moro, Stefano; Spalluto, Giampiero
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