Sfoglia per Autore
Computational Design of New Cyclic Urea Inhibitors for Improved Binding of HIV-1 Aspartic Protease.
2000-01-01 Kotamarthi, B.; Bonin, I.; Benedetti, Fabio; Miertus, S.
Facile inversion of configuration of N-Boc-b-aminoalcohols via SN2 cyclization to oxazolidinones.
2000-01-01 Benedetti, Fabio; Norbedo, S.
Pure homo-bifunctional poly(ethylene glycol) orthogonally protected: synthesis and characterisation
2001-01-01 Drioli, Sara; Benedetti, Fabio; Bonora, Gm
A study of the molecular structure and spectroscopic properties of polycyclic polyaza-compounds with diamond lattice
2001-01-01 Galasso, Vinicio; Benedetti, Fabio; Jones, D; Modelli, A.
Antibody Catalyzed Modification of Aminoacids. Efficient Hydrolysis of Tyrosine Benzoate.
2001-01-01 Benedetti, Fabio; Berti, Federico; Colombatti, A.; Flego, Massimiliano; Gardossi, Lucia; Linda, Paolo; Peressini, Silvia
Synthesis of all stereoisomers of cognac lactones via microbial reduction and enzymatic resolution strategies
2001-01-01 Forzato, Cristina; Benedetti, Fabio; Nitti, Patrizia; Pitacco, Giuliana; Valentin, Ennio; M., Vicario
Cyclic nitronic esters from highly diastereoselective cycloaddition of 2-(4-morpholinyl)norbornene to conjugated nitroolefins.
2001-01-01 Benedetti, Fabio; Drioli, Sara; Nitti, Patrizia; Pitacco, Giuliana; Valentin, Ennio
C2-Symmetric Val-Val dipeptide isosteres via diethylaluminium azide ring opening of epoxyalcohols.
2001-01-01 Benedetti, Fabio; Miertus, S.; Norbedo, S.
Epoxyalcohol route to hydroxyethylene dipeptide isosteres: a new synthesis of the diaminoalcohol core of HIV-protease inhibitor ABT-538 (ritonavir).
2001-01-01 Benedetti, Fabio; Norbedo, S.
Epoxyalcohol Route to Hydroxyethylene Dipeptide Isosteres. Stereodivergent Synthesis of the Diaminoalcohol Core of Ritonavir and its C-2 Epimer.
2002-01-01 Benedetti, Fabio; Berti, Federico; Norbedo, Stefano
GRID / tetrahedral intermediate computational approach to the study of selectivity of penicillin G acylase in amide bond synthesis
2002-01-01 Basso, A; Braiuca, Paolo; Ebert, Cynthia; Gardossi, Lucia; Linda, Paolo; Benedetti, Fabio
Albumin-controlled stereoselective reduction of 1,3-diketones to anti-diols
2002-01-01 Benedetti, Fabio; Berti, Federico; Donati, Ivan; Fregonese, Massimo
Design, synthesis and preliminary evaluation of peptidomimetic inhibitors of HIV aspartic protease with an epoxyalcohol core
2003-01-01 Benedetti, Fabio; Berti, Federico; Miertus, S.; Romeo, Domenico; Schillani, F.; Tossi, Alessandro
Small hydroxyethylene-based peptidomimetics inhibiting both HIV-1 and C. albicans aspartic protease
2003-01-01 Tossi, Alessandro; Benedetti, Fabio; Norbedo, Stefano; Skrbec, D.; Berti, Federico; Romeo, Domenico
Unexpected 1,2,3-triazole formation in the reaction of diethylaluminum azide with a’- amino a,b-unsaturated ketones.
2003-01-01 Adamo, I.; Benedetti, Fabio; Berti, Federico; Nardin, G.; Norbedo, S.
Val-Ala Dipeptide Isosteres via Hydrocyanation of alfa'-Amino-alfa,beta-Unsaturated Ketones. Control of Stereoselectivity by the N-Protecting Group.
2003-01-01 Benedetti, Fabio; Berti, Federico; Garau, G.; Martinuzzi, I.; Norbedo, S.
A Catalytic Antibody Programmed for Torsional Activation of Amide Bond Hydrolysis
2003-01-01 Aggarwal, R.; Benedetti, Fabio; Berti, Federico; Buchini, Sabrina; Colombatti, A.; Dinon, Francesca; Galasso, Vinicio; Norbedo, Stefano
Inibitori peptidomimetici di HIV-PR basati su isosteri diamminodiolici del dipeptide Phe-Pro
2004-01-01 Benedetti, Fabio; Berti, Federico; Campaner, Pietro; Dinon, Francesca; Tossi, Alessandro
An Unprecedented Catalytic Motif Revealed in The Model Structure of Amide Hydrolyzing Antibody 312D6.
2004-01-01 Benedetti, Fabio; Berti, Federico; Brady, K.; Colombatti, A.; Pauletto, A.; Pucillo, C.; Thomas, N. R.
Synthesis of a val-pro diaminodiol dipeptide isostere by epoxyamine cyclization
2004-01-01 Benedetti, Fabio; Berti, Federico; Dinon, Francesca; Nardin, Giorgio; Norbedo, Stefano
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