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Synthesis and biological evaluation of a new class of acyl derivatives of 3-amino-1-phenyl-4,5-dihydro-1H-pyrazol-5-one as potential dual cyclooxygenase (COX-1 and COX-2) and human lipoxygenase (5-LOX) inhibitors.
2005-01-01 Cusan, C.; Spalluto, Giampiero; Prato, Maurizio; Adams, M.; Bodensieck, A.; Bauer, R.; Tubaro, Aurelia; Bernardi, P.; DA ROS, Tatiana
Synthesis and biological evaluation of a new series of 1,2,4-Triazolo(1,5-a)-1,3,5-triazines as human A2A adenosine receptor antagonists with improved water solubility
2011-01-01 Federico, Stephanie; Paoletta, S.; Cheong, S. L.; Pastorin, G.; Cacciari, B.; Stragliotto, S.; Klotz, K. N.; Siegel, J.; Gao, Z. G.; Jacobson, K. A.; Moro, S.; Spalluto, Giampiero
Synthesis and biological evaluation of alpha-bromoacryloylamido indolyl pyridinyl propenones as potent apoptotic inducers in human leukaemia cells
2018-01-01 Romagnoli, Romeo; Prencipe, Filippo; Lopez-Cara, Luisa Carlota; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco
Synthesis and biological evaluation of new antitubulin agents containing 2-(3,4,5-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold
2020-01-01 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto
Synthesis and biological evaluation of new aryl-alkyl(alkenyl)-4-benzylpiperidines, novel Sigma Receptor (SR) modulators, as potential anticancer-agents
2016-01-01 Rui, Marta; Rossi, Daniela; Marra, Annamaria; Paolillo, Mayra; Schinelli, Sergio; Curti, Daniela; Tesei, Anna; Cortesi, Michela; Zamagni, Alice; Laurini, Erik; Pricl, Sabrina; Schepmann, Dirk; Wűnsch, Bernhard; Urban, Ernst; Pace, Vittorio; Collina, Simona
Synthesis and biological evaluation of new phenidone analogues as potential dual cyclooxygenase (COX-1 and COX-2) and human lipoxygenase (5-LOX) inhibitors
2005-01-01 Cusan, C.; Spalluto, Giampiero; Prato, Maurizio; Adams, M.; Bodensieck, A.; Bauer, R.; Tubaro, Aurelia; Bernardi, P.; DA ROS, Tatiana
Synthesis and biological evaluation of new simple indolic non peptidic HIV Protease inhibitors: The effect of different substitution patterns
2014-01-01 Bonini, C; Chiummiento, L.; Di Blasio, N.; Funicello, M.; Lupattelli, P.; Tramutola, F.; Berti, Federico; Ostric, Adrian; Miertus, S.; Frecer, V.; Kong, D. X.
Synthesis and biological evaluation of novel small non-peptidic HIV-1 PIs: The benzothiophene ring as an effective moiety
2012-01-01 Lucia, Chiummiento; Maria, Funicello; Paolo, Lupattelli; Francesco, Tramutola; Berti, Federico; Francesca Marino, Merlo
Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors
2015-01-01 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Prencipe, Filippo; Preti, Delia; Saponaro, Giulia; Romagnoli, Romeo; Gessi, Stefania; Merighi, Stefania; Stefanelli, Angela; Fazzi, Debora; Borea, Pier Andrea; Maia, Rodolfo C. outo; Romeiro, Nelilma C.; Fraga, Carlos A. M; Barreiro, Eliezer J.
Synthesis and Biological Properties of Fullerene-containing Amino Acids and Peptides
2004-01-01 D., Pantarotto; N., Tagmatarchis; A., Bianco; Prato, Maurizio
Synthesis and biological properties of new α-methylene-γ-butyrolactones and α,β-unsaturated δ-lactones
2006-01-01 Cateni, Francesca; J., Zilic; Zacchigna, Marina; P., Bonivento; F., Frausin; Scarcia, Vito
SYNTHESIS AND BIOLOGICAL RESOLUTION OF CONDENSED BICYCLIC ISOPARACONIC ACID DERIVATIVES
2000-01-01 Valentin, Ennio; Drioli, Sara; Felluga, Fulvia; Forzato, Cristina; Pitacco, Giuliana
Synthesis and Biological Studies of a New Series of 5-Heteroarylcarbamoylaminopyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as Human A3 Adenosine Receptor Antagonists. Influence of the Heteroaryl Substituent on Binding Affinity and Molecular Modeling Investigations
2006-01-01 Pastorin, G; DA ROS, Tatiana; Bolcato, C; Montopoli, C; Moro, S; Cacciari, B; Baraldi, P. G.; Varani, K; Borea, P. A.; Spalluto, Giampiero
Synthesis and Catalytic Activity of Gold Nanoparticles Supported on Dendrimeric Nanocellulose Hybrids
2016-01-01 HERREROS LOPEZ, ANA MARIA; A. AHAD HADAD, Caroline; Yate, Luis; Alshatwi, Ali A.; Vicentini, Nicola; Carofiglio, Tommaso; Prato, Maurizio
Synthesis and CD study of optically active bicyclic gamma-lactones belonging to the m-menthane series
1996-01-01 Forzato, Cristina; Nitti, Patrizia; Pitacco, Giuliana; Valentin, Ennio
Synthesis and characterisation of Cerium carbonate
1989-01-01 Lucchini, E; Schmid, Chiara
Synthesis and characterization of [pyRh(salen)adam], an adamantyl Rh-III complex containing bis(salicylaldehyde)ethylendiiminate as equatorial ligand
1995-01-01 Dreos, Renata; Geremia, Silvano; Randaccio, L.; Ruffini, S.; Tauzher, G.
Synthesis and characterization of a carbon nanotube-dendron series for efficient siRNA delivery
2009-01-01 Herrero M. A., Toma F. M.; Al Jamal, K. T.; Kostarelos, K.; Bianco, A.; DA ROS, Tatiana; Bano, F.; Casalis, L.; Scoles, G.; Prato, Maurizio
Synthesis and characterization of a diruthenium(II,III)-ketoprofen compound and study of the in vitro effects on CRC cells in comparison to the naproxen and ibuprofen derivatives
2012-01-01 Santos, Rlsr; Bergamo, Alberta; Sava, Gianni; De Oliveira Silva, D.
Synthesis and characterization of a hydrophilic conjugated 4+4 Re(I)-porphyrin metallacycle
2016-01-01 Milano, Domenico; Đorđević, Luka; Zangrando, Ennio; Iengo, Elisabetta; Tecilla, Paolo
SYNTHESIS AND CHARACTERIZATION OF A NOVEL GLYCOPOLYMER WITH PROTECTIVE ACTIVITY TOWARD HUMAN ANTI-ALFA-GAL ANTIBODIES
2002-01-01 Vetere, Amedeo; Donati, I.; Campa, C.; Semeraro, Sabrina; Gamini, Amelia; Paoletti, Sergio
Synthesis and Characterization of a Novel Glycopolymer with Protective Activity Toward Human Anti-α-Gal antibodies
2002-01-01 Vetere, A; Donati, Ivan; Campa, C; Semeraro, Sabrina; Gamini, Amelia; Paoletti, Sergio
Synthesis and characterization of a novel tetranuclear bimetallic complex containing rhodium(II) and zinc(II) as metal centres
1995-01-01 Maria, Kubiak; Tadeusz, Głowiak; Monika, Moszner; Jésef J., Ziółkowski; Asaro, Fioretta; Giacomo, Costa; Giorgio, Pellizer; Tavagnacco, Claudio
Synthesis and Characterization of Both Enantiomers of a Chiral C60 Derivative with C2 Symmetry
1995-01-01 M., Maggini; A., Bianco; G., Scorrano; C., Toniolo; Prato, Maurizio
Synthesis and characterization of constitutionally isomeric oriented calix[6]arene-based rotaxanes
2016-01-01 Zanichelli, V.; Ragazzon, G.; Arduini, A.; Credi, A.; Franchi, P.; Orlandini, G.; Venturi, M.; Lucarini, M.; Secchi, A.; Silvi, S.
Synthesis and Characterization of Highly Water-Soluble Dendrofulleropyrrolidine Bisadducts with DNA Binding Activity
2012-01-01 Montellano Lopez, A.; Scarel, F.; Rubio Carrero, N.; Vàzquez, E.; DA ROS, Tatiana; Prato, Maurizio
Synthesis and Characterization of Isomeric Binuclear Double- Bridged Alkylidene Tetraphenyldiphosphine and Diphenylphosphido Methylenediphenylphosphine Iron Nitrosyl Complexes
1987-01-01 Chau, C. N.; Yu, Y. F.; Wojcicki, A.; Calligaris, Mario; Nardin, Giorgio; Balducci, Gabriele
Synthesis and characterization of monochelated carboxylato palladium(II) complexes with nitrogen-donor chelating ligands. Crystal structures of diacetato(1,10-phenanthroline)palladium(II) and diacetato(2,9-dimethyl-1,10-phenanthroline)palladium(II)
1994-01-01 Milani, Barbara; Alessio, Enzo; Mestroni, Giovanni; Sommazzi, A.; Garbassi, F.; Zangrando, Ennio; BRESCIANI PAHOR, N.; Randaccio, L.
Synthesis and characterization of monochelated carboxylatopalladium(II) complexes with nitrogen-donor chelating ligands. Crystal structures of diacetato(1,10-phenanthroline)- and diacetato(2,9-dimethyl-1,10-phenanthroline)-palladium(II)
1994-01-01 Milani, B.; Alessio, E.; Mestroni, G.; Sommazzi, A.; Garbassi, F.; Zangrando, E.; Bresciani-Pahor, N.; Randaccio, L.
Synthesis and characterization of new chiral P,O ferrocenyl ligands and catalytic application to asymmetric Suzuki-Miyaura coupling
2014-01-01 Bayda, Samer; Cassen, Audrey; Daran, Jean Claude; Audin, Catherine; Poli, Rinaldo; Manoury, Eric; Deydier, Eric
Synthesis and characterization of new halogen -tetramethylene sulfoxide-ruthenium(II) and ruthenium(III) complexes; crystal structure of cis-dichlorotetrakis(tetramethylene sulfoxide) ruthenium(II) and hydrogen trans-bis(tetramethylene sulfoxide)tetrachlororuthenate(III)
1990-01-01 Alessio, Enzo; Milani, Barbara; G., Mestroni; M., Calligaris; P., Faleschini; W. M., Attia
Synthesis and characterization of new multifunctional high-molecular weight PEG derivatives (MultiPEG)s
2008-01-01 Drioli, S; Bonora, GIAN MARIA; Ballico, M.
Synthesis and characterization of new multifunctional self-boosted filters for UV protection: ZnO complex with dihydroxyphenyl benzimidazole carboxylic acid
2019-01-01 Battistin, M.; Durini, E.; Dissette, V.; Bonetto, A.; Marcomini, A.; Casagrande, E.; Brunetta, A.; Ziosi, P.; Molesini, S.; Gavioli, R.; Nicoli, F.; Manfredini, S.; Vertuani, S.; Baldisserotto, A.
Synthesis and Characterization of Novel Nucleobase-Carbon Nanotube Hybrids
2009-01-01 P., Singh; J., Kumar; F. M., Toma; J., Raya; Prato, Maurizio; B., Fabre; S., Verma; A., Bianco
Synthesis and characterization of palladacyclopentadiene complexes with N-heterocyclic carbene ligands
2015-01-01 Canovese, Luciano; Santo, Claudio; Scattolin, Thomas; Visentin, Fabiano; Bertolasi, Valerio
Synthesis and characterization of poly(3-alkylthiophenes) with NLO chromophoric groups in side chains
2002-01-01 Della Casa, Carlo; FRALEONI MORGERA, Alessandro; Costa Bizzarri, Paolo; Lanzi, Massimiliano; Paganin, Luisa
Synthesis and characterization of polyaspartamide copolymers obtained by ATRP for nucleic acid delivery
2014-01-01 G., Cavallaro; M., Licciardi; G., Amato; C., Sardo; G., Giammona; Farra, Rossella; Dapas, Barbara; Grassi, Mario; Grassi, Gabriele
Synthesis and characterization of polyglucuronan
1995-01-01 C., Bertocchi; P. A., Konowicz; S., Signore; F., Zanetti; A., Flaibani; Paoletti, Sergio; V., Crescenzi
Synthesis and Characterization of the First Fullerene-Peptide
1993-01-01 Prato, Maurizio; A., Bianco; M., Maggini; G., Scorrano; C., Toniolo; F., Wudl
Synthesis and characterization of trans-di-(4-pyridyl)porphyrin dimers
2016-01-01 Pisano, Simone; Milano, Domenico; Passoni, Nicola; Iengo, Elisabetta; Tecilla, Paolo
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