ArTS Archivio della ricerca di Trieste

BENEDETTI, FABIO
 Distribuzione geografica
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Continente #
NA - Nord America 7.469
EU - Europa 3.759
AS - Asia 969
SA - Sud America 17
AF - Africa 15
Continente sconosciuto - Info sul continente non disponibili 8
OC - Oceania 7
Totale 12.244
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Nazione #
US - Stati Uniti d'America 7.433
PL - Polonia 779
SE - Svezia 701
IT - Italia 648
UA - Ucraina 565
CN - Cina 420
TR - Turchia 216
DE - Germania 212
HK - Hong Kong 203
FI - Finlandia 190
GB - Regno Unito 171
BG - Bulgaria 111
IE - Irlanda 95
FR - Francia 94
CH - Svizzera 57
BE - Belgio 32
RU - Federazione Russa 30
CA - Canada 29
IN - India 29
ES - Italia 28
SG - Singapore 17
VN - Vietnam 15
SN - Senegal 13
KR - Corea 12
IR - Iran 11
NL - Olanda 10
BR - Brasile 8
EU - Europa 8
JP - Giappone 8
EE - Estonia 7
IL - Israele 7
MY - Malesia 7
RO - Romania 7
AU - Australia 6
ID - Indonesia 6
MX - Messico 5
PK - Pakistan 5
PH - Filippine 4
CL - Cile 3
NO - Norvegia 3
PT - Portogallo 3
RS - Serbia 3
BD - Bangladesh 2
CO - Colombia 2
CZ - Repubblica Ceca 2
HU - Ungheria 2
IQ - Iraq 2
LK - Sri Lanka 2
PE - Perù 2
SI - Slovenia 2
SK - Slovacchia (Repubblica Slovacca) 2
AR - Argentina 1
AZ - Azerbaigian 1
CI - Costa d'Avorio 1
CR - Costa Rica 1
DK - Danimarca 1
GR - Grecia 1
HR - Croazia 1
MD - Moldavia 1
ME - Montenegro 1
NG - Nigeria 1
NP - Nepal 1
NZ - Nuova Zelanda 1
PA - Panama 1
SA - Arabia Saudita 1
VE - Venezuela 1
Totale 12.244
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Città #
Woodbridge 1.008
Ann Arbor 896
Warsaw 779
Fairfield 769
Houston 738
Chandler 716
Jacksonville 501
Ashburn 448
Wilmington 404
Seattle 309
Cambridge 288
Hong Kong 202
Princeton 190
Izmir 189
Trieste 184
Beijing 117
Sofia 106
Dublin 95
Dearborn 92
Boardman 82
Bern 53
Milan 51
San Diego 45
Verona 36
Redwood City 34
Grafing 33
Des Moines 32
Bremen 30
Jinan 28
Düsseldorf 26
Brussels 25
Columbus 25
Chicago 24
Kocaeli 24
Mestre 23
Helsinki 22
Falls Church 21
Shenyang 21
Guangzhou 19
Nanjing 19
Norwalk 19
Fremont 17
London 17
Buffalo 16
Hefei 16
Phoenix 14
Auburn Hills 13
Dakar 13
Denton 13
Los Angeles 13
Ottawa 13
Washington 13
Dong Ket 12
Hebei 12
Kunming 12
Fuzhou 11
Hangzhou 11
Munich 11
Rome 11
Udine 11
Alcázar De San Juan 10
Toronto 10
Torre Del Greco 10
Tianjin 9
Venezia 9
Bologna 8
Changsha 8
Costa Mesa 8
Indiana 8
Sacile 8
Tallinn 7
Drancy 6
Mountain View 6
New York 6
Pune 6
Seoul 6
Shanghai 6
Andover 5
Ghent 5
Jerusalem 5
Redmond 5
San Francisco 5
Sevilla 5
Taizhou 5
Terni 5
Atlanta 4
Chengdu 4
Ciudad Real 4
Gorizia 4
Jakarta 4
Ningbo 4
Paris 4
St Louis 4
Zhengzhou 4
Assisi 3
Baotou 3
Belgrade 3
Caorle 3
Cuautitlán Izcalli 3
Detroit 3
Totale 9.197
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Nome #
Synthesis, characterization, and optimization for in vivo delivery of a nonselective isopeptidase inhibitor as new antineoplastic agent 360
The binding landscape of a partially-selective isopeptidase inhibitor with potent pro-death activity, based on the bis(arylidene)cyclohexanone scaffold 324
Synthesis of chiral, enantiopure allylic amines by the Julia olefination of α-amino esters 294
The isopeptidase inhibitor 2cPE triggers proteotoxic stress and ATM activation in chronic lymphocytic leukemia cells 289
1-Arylsulfonylamino-1,2,3-triazole derivatives from functionalized 1,2-cyclohexandiones 264
A Catalytic Antibody Programmed for Torsional Activation of Amide Bond Hydrolysis 243
Chlorogenic Compounds from Coffee Beans Exert Activity against Respiratory Viruses 222
Efficient Biginelli Synthesis of 2-Aminodihydropyrimidines under Microwave Irradiation 212
Strategies for delivery of siRNAs to ovarian cancer cells 208
Synthesis of a val-pro diaminodiol dipeptide isostere by epoxyamine cyclization 201
Fluorescent molecularly imprinted nanogels for the detection of anticancer drugs in human plasma 184
7-oxo-4,5,6,7-tetrahydroindole Derivatives from Nitro-olefins and Secondary a-keto enamines. 183
An Albumin-Derived Peptide Scaffold Capable of Binding and Catalysis 180
Activation parameters for intramolecular nucleophilic substitution by carbanions?the insignificant effect of ring strain on cyclisation rates 180
Development and evaluation of an immunoassay for the monitoring of the anti-HIV drug amprenavir 175
Stereoselective Hydroazidation of Amino Enones: Synthesis of the Ritonavir/Lopinavir Core 174
Synthesis and Biological Activity of Potent HIV-1 Protease Inhibitors Based on Phe-Pro Dihydroxyethylene Isosteres 170
A Competitive Immunoassay for the Detection of Esterolytic Activity of Antibodies and Enzymes 167
Aldolase Activity of Serum Albumins 162
1-Substituted morpholino ethenes—III. Carbocyclic and Aliphatic Heterocyclic Compounds from 5-Membered Ring Derivatives 161
An Enzyme-linked Immunosorbent Assay for the Direct Analysis of b-agonist Drugs in Urine and Sera 153
Structure Based Design of Inhibitors of Aspartic Protease of HIV-1 149
Versatile and stereoselective synthesis of diamino diol dipeptide isosteres, core units of pseudopeptide HIV protease inhibitors 149
Epoxyalcohol Route to Hydroxyethylene Dipeptide Isosteres. Stereodivergent Synthesis of the Diaminoalcohol Core of Ritonavir and its C-2 Epimer. 149
Nucleophilic addition to styryl sulphones. part II. Regio- and stereochemistry of the addition of enamines from 4-substituted cyclohexanones 148
The Non-Peptidic HIV Protease Inhibitor Tipranavir and Two Synthetic Peptidomimetics (TS98 and TS102) Modulate Pneumocystis carinii Growth and Proteasome Activity of HEL299 Cell Line 147
An Unprecedented Catalytic Motif Revealed in The Model Structure of Amide Hydrolyzing Antibody 312D6. 146
Synthesis of all stereoisomers of cognac lactones via microbial reduction and enzymatic resolution strategies 144
A potent HIV protease inhibitor identified in an epimeric mixture by high-resolution protein crystallography 144
Designing short peptides with high affinity for organic molecules: a combined docking, molecular dynamics and Monte Carlo approach 141
null 139
Reactivity of Cyclopentanone Enamines towards Acyl Aryldiazenes 138
Electron impact mass spectrometry of some geminal bis- sulphones 135
Impact of Stereochemistry on Ligand Binding: X-ray Crystallographic Analysis of an Epoxide-Based HIV Protease Inhibitor 134
Efficient Chemoenzymatic Synthesis of Chiral Pincer Ligands 133
Albumin-directed stereoselective reduction of 1,3-diketones and beta-hydroxyketones to anti diols 133
Intramolecular ring opening of epoxides by bis-activated carbanions. The influence of ring size on reactivity and selectivity 131
Modeling of Solvent Effects in the Activation of the Lipase from Rhizomucor Miehei 130
GRID / tetrahedral intermediate computational approach to the study of selectivity of penicillin G acylase in amide bond synthesis 130
Electron impact induced deamination of 1-sulphonylamino- 1,2,3-triazoles. 128
Addressing the poly- to oligo-ketone selectivity in styrene carbonylation catalyzed by Pd/bpy complexes. Effect of the 6-alkyl substitution 126
Synthesis and Biological Activity of New Mixed HIV-Pr Inhibitors Conjugated to Bifunctional High Molecular Weight poly(Ethylene)glycol 126
Regio- and Stereoselective Ring Opening of 2,3-Epoxyalcohols with Diethylaluminium Azide 125
Ring-Opening of Epoxyalcohols by Diethylaluminium Cyanide. Regio- and Stereoselective Synthesis of 1-Cyano-2,3-diols. 125
Chiral Pincer Ruthenium and Osmium Complexes for the Fast and Efficient Hydrogen Transfer Reduction of Ketones 122
Small hydroxyethylene-based peptidomimetics inhibiting both HIV-1 and C. albicans aspartic protease 121
Flexible synthesis of symmetric and non-symmetric hiv-1 protease inhibitors based on all-s-diaminodiol isosteres 118
Inibitori peptidomimetici di HIV-PR basati su isosteri diamminodiolici del dipeptide Phe-Pro 116
Reactivity of secondary functionalized enamines towards electrophilic diazenes. 116
E2F1 as a molecular drug target in ovarian cancer 115
Aspartic protease inhibitors. An integrated approach for the design and synthesis of diaminodiol based peptidomimetics 114
Epoxyalcohol route to hydroxyethylene dipeptide isosteres: a new synthesis of the diaminoalcohol core of HIV-protease inhibitor ABT-538 (ritonavir). 112
Computational Design of New Cyclic Urea Inhibitors for Improved Binding of HIV-1 Aspartic Protease. 112
Methyl effects in the cyclisation of g-epoxy bis-sulfones 112
Val-Ala Dipeptide Isosteres via Hydrocyanation of alfa'-Amino-alfa,beta-Unsaturated Ketones. Control of Stereoselectivity by the N-Protecting Group. 111
A study of the molecular structure and spectroscopic properties of polycyclic polyaza-compounds with diamond lattice 111
Cyclic nitronic esters from highly diastereoselective cycloaddition of 2-(4-morpholinyl)norbornene to conjugated nitroolefins. 108
Nucleophilic Additions to a,ß-Unsaturated Sulphones. Part III. Regiochemistry of the Reaction of (E)-Phenyl ß-Cyanovinyl Sulphone with Nitrogen, Oxygen and Carbon Nucleophiles 108
PEPTIDOMIMETIC INHIBITORS OF RETROVIRAL PROTEASES AND THEIR USE AS ANTIVIRALS 107
One Pot Synthesis of Micromolar BACE-1 Inhibitors Based on the Dihydropyrimidinone Scaffold and Their Thia and Imino Analogues 106
Anti-Sulphonamide Antibodies Catalyze the Hydrolysis of a Heterocyclic Amide 105
The base-catalysed cyclization of ω-epoxy 1,1-bis-sulfones. Reactivity snd selectivity as a function of ring size 105
null 105
Nucleophilic addition to styryl sulphones. Part I. A study on the regiochemistry 105
Regiospecificity in nucleophilic displacement of aromatic nitro-groups 105
Notizia. Strutture spaziali in natura. La proposta formativa di Scienze erogata nell’a. a. 2019-20 dal Polo di Trieste della Fondazione “I Lincei per la Scuola” 105
Nucleophilic Additions to a,ß-Unsaturated Sulphones. IV. Addition-Desulphonylation in the Reactions of Vinyl Sulphones Bearing a ß-Carbonyl Function 104
New synthesis of 5-amino-4-hydroxy-2,6-dimethylheptanoic acid, a hydroxyethylene isostere of the Val-Ala dipeptide 102
Crystallography as a tool to identify the best inhibitor in a complex mixture 100
Synthesis and biological evaluation in vitro and in mammalian cells of new heteroaryl carboxyamides as HIV-protease inhibitors 100
Stereoselective synthesis of non symetric dihydroxyethylene dipeptide isosteres via epoxyalcohols derived from α-amino acids 98
Synthesis and Antiviral Activity of Novel Adamantylpeptides 98
Facile inversion of configuration of N-Boc-b-aminoalcohols via SN2 cyclization to oxazolidinones. 97
Reactivity of secondary cross-conjugated ketoenamines towards electrophilic diazenes. 95
Application of an Enzyme Immunoassay for the Detection of the Anabolic Agents Zeranol and 19-Nortestosterone 94
Transition States in Intramolecular SN2 Reactions of Carbanions. The Closure of 3-, 4- and 5-Membered Rings 94
Unexpected 1,2,3-triazole formation in the reaction of diethylaluminum azide with a’- amino a,b-unsaturated ketones. 93
Biocrystallographic study on drug resistant variants of HIV protease with new inhibitors 92
Pure homo-bifunctional poly(ethylene glycol) orthogonally protected: synthesis and characterisation 90
Carbon-13 N.m.r. Spectra of 1,1-Bis-Sulphones: ß-Effects and Conformation. 84
Albumin-controlled stereoselective reduction of 1,3-diketones to anti-diols 83
Cyclization of gamma-delta-Epoxy-alfa-cyanosulfones. A Simple, DiastereoselectiveRoute to Cyclopropane Carboxylic Acids. 80
l-Substituted morpholino ethenes. III. Carbocyclic and aliphatic heterocyclic compounds from 5-membered ring derivatives 79
DESIGN OF PEPTIDOMIMETIC INHIBITORS OF ASPARTIC PROTEASE OF HIV-1 CONTAINING -PHEpsiPRO- CORE AND DISPLAYING FAVOURABLE ADME-RELATED PROPERTIES 78
Enhancing proteotoxic stress in leiomyosarcoma cells triggers mitochondrial dysfunctions, cell death, and antitumor activity in vivo 78
Biocrystallographic study on drug resistant variants of HIV protease with new inhibitors 77
null 76
Effect of 6-alkyl substituted 2,2'-bipyridines in the Pd-catalyzed styrene carbonylation: shifting the selectivity from polyketones to oligoketones 76
Reactivity of phenylcarbamoyldiazene towards 1- aminocyclopentenes. 68
CADD of New Pseudopeptide Inhibitors of HIV-1 Aspartic Protease 67
Spatial and temporal patterns of nutrients distribution in the Ross Sea. 60
C2-Symmetric Val-Val dipeptide isosteres via diethylaluminium azide ring opening of epoxyalcohols. 58
Nutrient Utilization and Particulate Organic Matter Change in the Upper Mixed Layer (Ross Sea, Antarctica) 56
Stereoselective Synthesis of non Symmetric Dihydroxyethylene Dipeptide Isosteres via Epoxyalcohols Derived from alpha-Amino Acids 53
Elimination and addition reactions. Part 40. The insignificant effect of strain in higher order eliminations in 1,1-bis(phenylsulphonyl) carbanions with w-leaving groups 51
Antibody Catalyzed Modification of Aminoacids. Efficient Hydrolysis of Tyrosine Benzoate. 43
Design, synthesis and preliminary evaluation of peptidomimetic inhibitors of HIV aspartic protease with an epoxyalcohol core 29
Purification and Characterization of L,(L/D)-aminopeptidase from Guinea Pig Serum 24
Identification and evaluation of antiviral activity of novel compounds targeting SARS-CoV-2 virus by enzymatic and antiviral assays, and computational analysis 13
Totale 12.585
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Categoria #
all - tutte 29.035
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 29.035
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019708 0 0 0 0 0 0 0 0 0 0 498 210
2019/20202.279 134 92 116 398 152 311 265 259 177 138 162 75
2020/20211.823 152 105 173 242 148 171 75 141 149 208 86 173
2021/20221.391 50 94 90 160 31 113 58 38 155 151 110 341
2022/20231.895 198 265 171 258 196 323 7 149 212 15 68 33
2023/2024847 101 33 67 94 80 77 173 187 11 15 9 0
Totale 12.585